[3H]diprenorphine [Ligand Id: 1612] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • δ receptor in Human [GtoPdb: 317] [UniProtKB: P41143]
There should be some charts here, you may need to enable JavaScript!
  • κ receptor in Human [GtoPdb: 318] [UniProtKB: P41145]
There should be some charts here, you may need to enable JavaScript!
  • μ receptor in Mouse [GtoPdb: 319] [UniProtKB: P42866]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
δ receptor in Human [GtoPdb: 317] [UniProtKB: P41143]
GtoPdb - - 9.3 pKi 0.5 nM Ki NIDA Res Monogr (1998) 178: 440-66 [PMID:9686407];
J Biol Chem (1992) 267: 7921-6 [PMID:1313812]
κ receptor in Human [GtoPdb: 318] [UniProtKB: P41145]
GtoPdb - - 9.1 pKd 0.79 nM Kd Proc Natl Acad Sci USA (1995) 92: 7006-10 [PMID:7624359];
J Biol Chem (1992) 267: 7921-6 [PMID:1313812]
μ receptor in Mouse [GtoPdb: 319] [UniProtKB: P42866]
GtoPdb - - 10.1 pKd 0.08 nM Kd Mol Pharmacol (1994) 45: 330-4 [PMID:8114680]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.