TP-472 [Ligand Id: 9522] activity data from GtoPdb

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  • bromodomain containing 7 in Human [GtoPdb: 2726] [UniProtKB: Q9NPI1]
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  • bromodomain containing 9 in Human [GtoPdb: 2728] [UniProtKB: Q9H8M2]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
bromodomain containing 7 in Human [GtoPdb: 2726] [UniProtKB: Q9NPI1]
GtoPdb By isothermal titration calorimetry (ITC). - 6.47 pIC50 340 nM IC50 TP-472 A BRD9/7 Probe. Structural Genomics Consortium.
bromodomain containing 9 in Human [GtoPdb: 2728] [UniProtKB: Q9H8M2]
GtoPdb By isothermal titration calorimetry. - 7.48 pIC50 33 nM IC50 TP-472 A BRD9/7 Probe. Structural Genomics Consortium.

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.