OF-1 [Ligand Id: 9523] activity data from GtoPdb

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  • bromodomain and PHD finger containing 1 in Human [GtoPdb: 2730] [UniProtKB: P55201]
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  • bromodomain and PHD finger containing 3 in Human [GtoPdb: 2731] [UniProtKB: Q9ULD4]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
bromodomain and PHD finger containing 1 in Human [GtoPdb: 2730] [UniProtKB: P55201]
GtoPdb By isothermal titration calorimetry, using the BRPF1B isoform. - 7 pKd 100 nM Kd OF-1 A chemical probe for BRPF bromodomains. SGC
bromodomain and PHD finger containing 3 in Human [GtoPdb: 2731] [UniProtKB: Q9ULD4]
GtoPdb By isothermal titration calorimetry. - 5.62 pKd 2400 nM Kd OF-1 A chemical probe for BRPF bromodomains. SGC

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.