Ligand id: 9119

Name: BAY1238097

Compound class Synthetic organic
BAY 1238097 | BAY-1238097
Database Links
GtoPdb PubChem SID 315661204
BAY1238097 is a BET inhibitor. BET inhibitors bind to the bromodomains of the bromodomain and extra-terminal motif (BET) proteins BRD2, BRD3, BRD4, and BRDT. This mechanism acts to prevent protein-protein interaction between BET proteins and acetylated histones and transcription factors. The action disrupts chromatin remodeling and inhibits expression of some growth-promoting genes which slows proliferation in susceptible tumours.
The chemical structure for BAY1238097 has not been disclosed. We will present the structure upon its disclosure.