Ligand id: 9119

Name: BAY1238097

Compound class Synthetic organic
BAY 1238097 | BAY-1238097
BAY1238097 is a BET inhibitor. BET inhibitors bind to the bromodomains of the bromodomain and extra-terminal motif (BET) proteins BRD2, BRD3, BRD4, and BRDT. This mechanism acts to prevent protein-protein interaction between BET proteins and acetylated histones and transcription factors. The action disrupts chromatin remodeling and inhibits expression of some growth-promoting genes which slows proliferation in susceptible tumours.
The chemical structure for BAY1238097 has not been disclosed. We will present the structure upon its disclosure.
Database Links
GtoPdb PubChem SID 315661204