Compound class:
Synthetic organic
Comment: TAK-071 is a muscarinic M1 receptor positive allosteric modulator [1-2]. It has been shown to improve cognitive function in in vivo models.
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Bioactivity Comments |
TAK-071 has a relatively low α (cooperativity)-value (199) which reduces its propensity to induce cholinergic-mediated adverse gastrointestinal effects (diarrhea) [2]. |