Synonyms: ACT-539313 | ACT539313
Compound class:
Synthetic organic
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Bioactivity Comments |
Apparent equilibrium dissociation constant (Kb) for ACT‐539313 is 0.69 nM vs. OX1 and 42 nM vs. OX2 [1]. Its potency at non-human mammalian orexin receptors is similar to its potency at the human receptors. |