Synonyms: Ariane® | example 44 [WO2014036897A1] | SHR-3680 | SHR3680
rezvilutamide is an approved drug (China NMPA (2022))
Compound class:
Synthetic organic
Comment: Rezvilutamide is an oral, nonsteroidal androgen receptor antagonist [3].
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Bioactivity Comments |
Rezvilutamide inhibits testosterone-induced PSA secretion by LnCAP cells with an IC50 of 22nM in vitro, and inhibits LnCAP proliferation (IC50 33 nM) [3]. |