hsp90α1   Click here for help

GtoPdb Ligand ID: 7752

Synonyms: HSP90A | HSPC1 | HSPCA
Compound class: Endogenous peptide in human, mouse or rat
Species: Human
Other ligands which bind to or alter the activity of this ligand
Key to terms and symbols Click column headers to sort
Ligand Sp. Type Action Value Parameter Concentration range (M) Reference
pimitespib Small molecule or natural product Hs Inhibitor Inhibition 7.2 pIC50 - 2
⤷ pIC50 7.2 (IC50 6.9x10-8 M) [2]
Description: Competitive displacement of biotin-labeled geldanamycin from immobilised His-tagged HSP90α N terminal domain using an AlphaScreen assay.
tanespimycin Small molecule or natural product Primary target of this compound Hs Inhibitor Inhibition 6.1 pIC50 - 1
⤷ pIC50 6.1 (IC50 7.8x10-7 M) [1]
Description: fluorescence polarization assay