Synonyms: CGP 13501 | CGP-13501
Compound class:
Synthetic organic
Comment: CGP13501 is a positive allosteric modulator of GABAB Class C GPCRs [1] which potentiates GABA-induced GTPγ[35S] binding, but displays no intrinsic agonist activity.
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Bioactivity Comments |
CGP13501 significantly increases GABA-induced GTP&gamma'[35S] binding to CHO cell membranes containing human GABAB1 and rat GABAB2 subunits [1]. |