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Compound class:
Synthetic organic
Comment: Bromosporine is a broad spectrum inhibitor of bromodomain-containing proteins. This is contained in the Structural Genomics Consortium's (SGC) Epigenetics Probes Collection.
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Bioactivity Comments |
Differential scanning fluorimetry (DSF) data on the Structural Genomics Consortium's (SGC) website indicates that bromosporine inhibits BRD-containing proteins including BRD2, BRD3, BRD4, BRD9, BRDT and CECR2 [1]. |