Ligand id: 7129

Name: bisoprolol

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Structure and Physico-chemical Properties

2D Structure
Calculated Physico-chemical Properties
Hydrogen bond acceptors 4
Hydrogen bond donors 2
Rotatable bonds 12
Topological polar surface area 59.95
Molecular weight 325.23
XLogP 2.37
No. Lipinski's rules broken 1

Molecular properties generated using the CDK

No information available.
Summary of Clinical Use
Used to treat hypertension, stable chronic angina and specific forms of stable chronic heart failure.
Mechanism Of Action and Pharmacodynamic Effects
Bisoprolol blocks catecholamine stimulation of β1-adrenoceptors in the heart to lower the heart rate and blood pressure.
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