[125I]Tyr3 SMS 201-995   Click here for help

GtoPdb Ligand ID: 2062

Synonyms: [125I][Tyr3]octreotide
 Ligand is labelled  Ligand is radioactive
Compound class: Peptide or derivative
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Ligand Activity Visualisation Charts

These are box plot that provide a unique visualisation, summarising all the activity data for a ligand taken from ChEMBL and GtoPdb across multiple targets and species. Click on a plot to see the median, interquartile range, low and high data points. A value of zero indicates that no data are available. A separate chart is created for each target, and where possible the algorithm tries to merge ChEMBL and GtoPdb targets by matching them on name and UniProt accession, for each available species. However, please note that inconsistency in naming of targets may lead to data for the same target being reported across multiple charts.

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View interactive charts of activity data across species
References
1. Feuerbach D, Fehlmann D, Nunn C, Siehler S, Langenegger D, Bouhelal R, Seuwen K, Hoyer D. (2000)
Cloning, expression and pharmacological characterisation of the mouse somatostatin sst(5) receptor.
Neuropharmacology, 39 (8): 1451-62. [PMID:10818261]
2. Reubi JC. (1985)
New specific radioligand for one subpopulation of brain somatostatin receptors.
Life Sci, 36 (19): 1829-36. [PMID:2859510]
3. Siehler S, Seuwen K, Hoyer D. (1998)
[125I][Tyr3]octreotide labels human somatostatin sst2 and sst5 receptors.
Eur J Pharmacol, 348 (2-3): 311-20. [PMID:9652348]
4. Siehler S, Seuwen K, Hoyer D. (1999)
Characterisation of human recombinant somatostatin receptors. 1. Radioligand binding studies.
Naunyn Schmiedebergs Arch Pharmacol, 360 (5): 488-99. [PMID:10598788]
5. Wester HJ, Schottelius M, Scheidhauer K, Reubi JC, Wolf I, Schwaiger M. (2002)
Comparison of radioiodinated TOC, TOCA and Mtr-TOCA: the effect of carbohydration on the pharmacokinetics.
Eur J Nucl Med Mol Imaging, 29 (1): 28-38. [PMID:11807604]