kallikrein 1

Target id: 2865

Nomenclature: kallikrein 1

Family: S1: Chymotrypsin

Annotation status:  image of a grey circle Awaiting annotation/under development. Please contact us if you can help with annotation.  » Email us

   GtoImmuPdb view: OFF :     Currently no data for kallikrein 1 in GtoImmuPdb

Gene and Protein Information
Species TM AA Chromosomal Location Gene Symbol Gene Name Reference
Human - 262 19q13.3 KLK1 kallikrein 1
Mouse - 261 7 B4 Klk1 kallikrein 1
Rat - 265 1q22 Klk1 kallikrein 1
Previous and Unofficial Names
renal/pancreas/salivary kallikrein
Database Links
Specialist databases
MEROPS S01.160 (Hs)
Other databases
BRENDA
ChEMBL Target
Ensembl Gene
Entrez Gene
GenitoUrinary Development Molecular Anatomy Project
Human Protein Atlas
KEGG Enzyme
KEGG Gene
OMIM
RefSeq Nucleotide
RefSeq Protein
UniProtKB
Wikipedia
Enzyme Reaction
EC Number: 3.4.21.35

Download all structure-activity data for this target as a CSV file

Inhibitors
Key to terms and symbols View all chemical structures Click column headers to sort
Ligand Sp. Action Affinity Units Reference
example 131 [WO2009133348] Hs Inhibition 9.3 pIC50 1
pIC50 9.3 (IC50 5.4x10-10 M) [1]

References

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1. Evans DM, Allan CE, Horton J, Rooker DP. (2009) Aminopyridine derivatives. Patent number: WO2009133348. Assignee: Vantia Limited.. Priority date: 29/04/2008. Publication date: 05/11/2009.

How to cite this page

S1: Chymotrypsin: kallikrein 1. Last modified on 22/09/2015. Accessed on 11/12/2017. IUPHAR/BPS Guide to PHARMACOLOGY, http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=2865.