GluK5 | Ionotropic glutamate receptors | IUPHAR/BPS Guide to PHARMACOLOGY

Top ▲

GluK5

Target not currently curated in GtoImmuPdb

Target id: 454

Nomenclature: GluK5

Family: Ionotropic glutamate receptors

Annotation status:  image of a grey circle Awaiting annotation/under development. Please contact us if you can help with annotation.  » Email us

Gene and Protein Information
Species TM P Loops AA Chromosomal Location Gene Symbol Gene Name Reference
Human 3 1 980 19q13.2 GRIK5 glutamate ionotropic receptor kainate type subunit 5
Mouse 3 1 979 7 A3 Grik5 glutamate receptor
Rat 3 1 979 1q21 Grik5 glutamate ionotropic receptor kainate type subunit 5
Previous and Unofficial Names
GRIK2 | glutamate receptor KA2 | GluRgamma2 | EAA2 | GLUK2 | glutamate receptor, ionotropic, kainate 5 | glutamate receptor, ionotropic, kainate 5 (gamma 2) | glutamate receptor
Database Links
ChEMBL Target
Ensembl Gene
Entrez Gene
Human Protein Atlas
KEGG Gene
OMIM
RefSeq Nucleotide
RefSeq Protein
UniProtKB
Wikipedia
Natural/Endogenous Ligands
L-glutamic acid

Download all structure-activity data for this target as a CSV file

Agonists
Key to terms and symbols View all chemical structures Click column headers to sort
Ligand Sp. Action Affinity Parameter Reference
[3H]SYM2081 Hs Full agonist - -
[3H]kainate Hs Full agonist - -
domoic acid Hs Full agonist - -
dysiherbaine Hs Full agonist - -
kainate Hs Full agonist - -
SYM2081 Hs Full agonist - -

Contributors

Show »

How to cite this page

Bernhard Bettler, Graham L. Collingridge, Ray Dingledine, Stephen F. Heinemann, Michael Hollmann, Juan Lerma, David Lodge, Mark Mayer, Masayoshi Mishina, Christophe Mulle, Shigetada Nakanishi, Richard Olsen, Stephane Peineau, John A. Peters, Peter Seeburg, Michael Spedding, Jeffrey C. Watkins, Robert J. Wenthold.
Ionotropic glutamate receptors: GluK5. Last modified on 20/10/2015. Accessed on 20/02/2019. IUPHAR/BPS Guide to PHARMACOLOGY, http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=454.