Synonyms: 4306 CB | Tranxene®
clorazepate is an approved drug (FDA (1972))
Compound class:
Synthetic organic
Comment: The marketed formulation is a racemic mixture of stereo-isomers; R-clorazepate and S-clorazepate. We show the non-isomeric molecule to represent this mixture.
|
|
Bioactivity Comments |
Clorazepate positively modulates the activity of GABAA receptors expressed in Xenopus oocytes injected with chick embryo mRNA, with a Ki of 390nM [1]. There appears to be no publicly available bioactivity data for this drug at its human molecular target so we have not mapped a primary drug target in this instance. |