Ligand id: 4818

Name: tiagabine

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Structure and Physico-chemical Properties

2D Structure
Calculated Physico-chemical Properties
Hydrogen bond acceptors 3
Hydrogen bond donors 1
Rotatable bonds 6
Topological polar surface area 97.02
Molecular weight 375.13
XLogP 4.01
No. Lipinski's rules broken 0

Molecular properties generated using the CDK

No information available.
Summary of Clinical Use
Tiagabine is an anticonvulsant medication used in the treatment of partial seizures and as an adjunctive treatment for epilepsy.
Mechanism Of Action and Pharmacodynamic Effects
The exact mechanism of action of tiagabine is unknown, however it is believed to operate as a selective GABA reuptake inhibitor.
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