azelastine

Ligand id: 7121

Name: azelastine

Structure and Physico-chemical Properties

2D Structure
Calculated Physico-chemical Properties
Hydrogen bond acceptors 4
Hydrogen bond donors 0
Rotatable bonds 3
Topological polar surface area 23.55
Molecular weight 381.16
XLogP 5.37
No. Lipinski's rules broken 1

Molecular properties generated using the CDK

No information available.
Summary of Clinical Use
Used to treat occular and nasal symptoms of hay fever and allergic conjunctivitis.
Mechanism Of Action and Pharmacodynamic Effects
Azelastine blocks the action of endogenous histamine at the histamine H1 receptor.
External links