Available chemical structures for ALK receptor tyrosine kinase inhibitors

ceritinib
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Targets
ALK receptor tyrosine kinase; Insulin receptor; Insulin-like growth factor I receptor; fms related receptor tyrosine kinase 3; testis specific serine kinase 1B
ensartinib
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Targets
ALK receptor tyrosine kinase; MET proto-oncogene, receptor tyrosine kinase
brigatinib
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Targets
ALK receptor tyrosine kinase; Insulin receptor; Insulin-like growth factor I receptor; epidermal growth factor receptor
GSK-1838705A
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Targets
ALK receptor tyrosine kinase; Insulin receptor; Insulin-like growth factor I receptor; ribosomal protein S6 kinase A1
gilteritinib
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Targets
ALK receptor tyrosine kinase; AXL receptor tyrosine kinase; MER proto-oncogene, tyrosine kinase; c-ros oncogene 1, receptor tyrosine kinase; fms related receptor tyrosine kinase 3; leukocyte receptor tyrosine kinase; neurotrophic receptor tyrosine kinase 1; ret proto-oncogene
TL13-112
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Targets
ALK receptor tyrosine kinase
compound 8e [PMID: 24432909]
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Targets
ALK receptor tyrosine kinase; FER tyrosine kinase; FES proto-oncogene, tyrosine kinase; c-ros oncogene 1, receptor tyrosine kinase; leukocyte receptor tyrosine kinase; mitogen-activated protein kinase kinase kinase 9; neurotrophic receptor tyrosine kinase 2
crizotinib
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Targets
ALK receptor tyrosine kinase; MET proto-oncogene, receptor tyrosine kinase
ficonalkib
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Targets
ALK receptor tyrosine kinase
neladalkib
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Targets
ALK receptor tyrosine kinase
repotrectinib
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Targets
ALK receptor tyrosine kinase; Janus kinase 2; c-ros oncogene 1, receptor tyrosine kinase; neurotrophic receptor tyrosine kinase 1; neurotrophic receptor tyrosine kinase 2; neurotrophic receptor tyrosine kinase 3
zotizalkib
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Targets
ALK receptor tyrosine kinase
dirozalkib
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Targets
ALK receptor tyrosine kinase
alectinib
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Targets
ALK receptor tyrosine kinase; MET proto-oncogene, receptor tyrosine kinase
compound 25b [PMID: 22564207]
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Targets
ALK receptor tyrosine kinase; FER tyrosine kinase; FES proto-oncogene, tyrosine kinase; NUAK family kinase 1; checkpoint kinase 2; ribosomal protein S6 kinase A2; ribosomal protein S6 kinase A3; ribosomal protein S6 kinase A6
envonalkib
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Targets
ALK receptor tyrosine kinase
CEP-37440
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Targets
ALK receptor tyrosine kinase; protein tyrosine kinase 2
AZD3463
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Targets
ALK receptor tyrosine kinase; Insulin-like growth factor I receptor
compound 5m [PMID: 20483621]
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Targets
ALK receptor tyrosine kinase; BMP2 inducible kinase
compound 5n [PMID: 20483621]
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Targets
ALK receptor tyrosine kinase; doublecortin like kinase 3; mitogen-activated protein kinase kinase kinase 3
iruplinalkib
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Targets
ALK receptor tyrosine kinase
compound 5g [PMID: 20483621]
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Targets
ALK receptor tyrosine kinase; doublecortin like kinase 1
compound 17 [PMID: 34176264]
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Targets
ALK receptor tyrosine kinase
compound 15 [PMID: 24900237]
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Targets
ALK receptor tyrosine kinase; Insulin receptor; unc-51 like kinase 3
unecritinib
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Targets
ALK receptor tyrosine kinase
belizatinib
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Targets
ALK receptor tyrosine kinase; AXL receptor tyrosine kinase; LCK proto-oncogene, Src family tyrosine kinase; MER proto-oncogene, tyrosine kinase; fms related receptor tyrosine kinase 3; interleukin 1 receptor associated kinase 1; leukocyte receptor tyrosine kinase; mitogen-activated protein kinase kinase kinase kinase 2
NVP-TAE684
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Targets
ALK receptor tyrosine kinase
lorlatinib
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Targets
ALK receptor tyrosine kinase; FES proto-oncogene, tyrosine kinase; c-ros oncogene 1, receptor tyrosine kinase

Please note that chemical structures may not be available for all inhibitors at this target. For more details please email us.