Available chemical structures for TEK receptor tyrosine kinase inhibitors

pexmetinib
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Targets
ABL proto-oncogene 1, non-receptor tyrosine kinase; ABL proto-oncogene 2, non-receptor tyrosine kinase; FYN proto-oncogene, Src family tyrosine kinase; HCK proto-oncogene, Src family tyrosine kinase; LYN proto-oncogene, Src family tyrosine kinase; TEK receptor tyrosine kinase; fibroblast growth factor receptor 1; fms related receptor tyrosine kinase 1; fms related receptor tyrosine kinase 4; misshapen like kinase 1; mitogen-activated protein kinase 11; mitogen-activated protein kinase 14
compound 8h [PMID: 21561767]
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Targets
ABL proto-oncogene 1, non-receptor tyrosine kinase; EPH receptor A2; EPH receptor A3; EPH receptor A7; TEK receptor tyrosine kinase; platelet derived growth factor receptor alpha; ret proto-oncogene
altiratinib
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Targets
MET proto-oncogene, receptor tyrosine kinase; TEK receptor tyrosine kinase; kinase insert domain receptor
merestinib
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Targets
AXL receptor tyrosine kinase; MER proto-oncogene, tyrosine kinase; MET proto-oncogene, receptor tyrosine kinase; TEK receptor tyrosine kinase; discoidin domain receptor tyrosine kinase 1; fms related receptor tyrosine kinase 3; macrophage stimulating 1 receptor; tyrosine kinase with immunoglobulin like and EGF like domains 1
CEP-11981
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Targets
BLK proto-oncogene, Src family tyrosine kinase; TEK receptor tyrosine kinase; fibroblast growth factor receptor 1; fms related receptor tyrosine kinase 1; kinase insert domain receptor; mitogen-activated protein kinase kinase kinase 7; neurotrophic receptor tyrosine kinase 1; neurotrophic receptor tyrosine kinase 2; ret proto-oncogene; serine/threonine kinase 3
linifanib
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Targets
KIT proto-oncogene, receptor tyrosine kinase; TEK receptor tyrosine kinase; colony stimulating factor 1 receptor; cyclin dependent kinase 19; cyclin dependent kinase 8; fms related receptor tyrosine kinase 1; fms related receptor tyrosine kinase 3; fms related receptor tyrosine kinase 4; kinase insert domain receptor; platelet derived growth factor receptor beta; ret proto-oncogene
compound 5 [PMID: 17618114]
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Targets
TEK receptor tyrosine kinase
compound 8i [PMID: 22765894]
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Targets
AXL receptor tyrosine kinase; KIT proto-oncogene, receptor tyrosine kinase; MET proto-oncogene, receptor tyrosine kinase; TEK receptor tyrosine kinase; fibroblast growth factor receptor 1; fms related receptor tyrosine kinase 1; fms related receptor tyrosine kinase 3; fms related receptor tyrosine kinase 4; kinase insert domain receptor; macrophage stimulating 1 receptor; platelet derived growth factor receptor alpha; platelet derived growth factor receptor beta
DDR1/2 inhibitor 5n
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Targets
ABL proto-oncogene 1, non-receptor tyrosine kinase; EPH receptor A2; EPH receptor A7; EPH receptor A8; EPH receptor B2; LCK proto-oncogene, Src family tyrosine kinase; TEK receptor tyrosine kinase; discoidin domain receptor tyrosine kinase 1; discoidin domain receptor tyrosine kinase 2; neurotrophic receptor tyrosine kinase 1; neurotrophic receptor tyrosine kinase 2; neurotrophic receptor tyrosine kinase 3; serine/threonine kinase 10

Please note that chemical structures may not be available for all inhibitors at this target. For more details please email us.