Available chemical structures for μ receptor antagonists

navacaprant
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Targets
δ receptor; κ receptor; μ receptor
[3H]diprenorphine
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Targets
δ receptor; κ receptor; μ receptor
[3H]naloxone
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Targets
μ receptor
naloxonazine
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Targets
μ receptor
samidorphan
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Targets
δ receptor; κ receptor; μ receptor
diprenorphine
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Targets
δ receptor; κ receptor; μ receptor
quadazocine
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Targets
δ receptor; κ receptor; μ receptor
(-)-bremazocine
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Targets
δ receptor; κ receptor; μ receptor
CTOP
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Targets
μ receptor
nalmefene
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Targets
δ receptor; κ receptor; μ receptor
β-FNA
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Targets
δ receptor; κ receptor; μ receptor
NFP
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Targets
δ receptor; κ receptor; μ receptor
naltrexone
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Targets
δ receptor; κ receptor; μ receptor
GSK1521498
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Targets
μ receptor
alvimopan
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Targets
δ receptor; κ receptor; μ receptor
levallorphan
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Targets
μ receptor
naloxone
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Targets
δ receptor; κ receptor; μ receptor
naldemedine
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Targets
δ receptor; μ receptor
nalorphine
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Targets
δ receptor; κ receptor; μ receptor
BNTX
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Targets
δ receptor; κ receptor; μ receptor
AT-076
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Targets
δ receptor; κ receptor; μ receptor; NOP receptor
methylnaltrexone
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Targets
δ receptor; κ receptor; μ receptor
CTAP
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Targets
δ receptor; μ receptor
naloxone benzoylhydrazone
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Targets
κ receptor; μ receptor
naltrindole
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Targets
δ receptor; κ receptor; μ receptor
naltriben
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Targets
δ receptor; κ receptor; μ receptor; TRPM7
nor-binaltorphimine
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Targets
δ receptor; κ receptor; μ receptor
aticaprant
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Targets
δ receptor; κ receptor; μ receptor
zyklophin
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Targets
δ receptor; κ receptor; μ receptor

Please note that chemical structures may not be available for all antagonists at this target. For more details please email us.