Available chemical structures for Estrogen receptor-α antagonists

norendoxifen
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Targets
CYP19A1; Estrogen receptor-α; Estrogen receptor-β
giredestrant
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Targets
Estrogen receptor-α
camizestrant
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Targets
Estrogen receptor-α
LSZ102
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Targets
Estrogen receptor-α
compound 5 [PMID: 40393772]
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Targets
Estrogen receptor-α
4-hydroxytamoxifen
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Targets
Estrogen receptor-α; Estrogen receptor-β; Estrogen-related receptor-γ; GPER
compound 17b [PMID: 35286086]
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Targets
Estrogen receptor-α; epidermal growth factor receptor
bazedoxifene
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Targets
Estrogen receptor-α; Estrogen receptor-β
GSK5182
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Targets
Estrogen receptor-α; Estrogen-related receptor-γ
hexestrol
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Targets
Estrogen receptor-α
imlunestrant
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Targets
Estrogen receptor-α
raloxifene
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Targets
Estrogen receptor-α; Estrogen receptor-β; GPER; aldehyde oxidase 1
fulvestrant
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Targets
Estrogen receptor-α; Estrogen receptor-β; GPER
clomiphene
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Targets
Estrogen receptor-α; VRAC
methyl-piperidino-pyrazole
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Targets
Estrogen receptor-α
tamoxifen
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Targets
CYP3A4; Estrogen receptor-α; Estrogen receptor-β; GPER; Maxi Cl-; VRAC
ospemifene
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Targets
Estrogen receptor-α; Estrogen receptor-β
ERD-308
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Targets
Estrogen receptor-α
amcenestrant
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Targets
Estrogen receptor-α

Please note that chemical structures may not be available for all antagonists at this target. For more details please email us.