Available chemical structures for Estrogen receptor-β antagonists

bazedoxifene
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Targets
Estrogen receptor-α; Estrogen receptor-β
4-hydroxytamoxifen
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Targets
Estrogen receptor-α; Estrogen receptor-β; Estrogen-related receptor-γ; GPER
fulvestrant
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Targets
Estrogen receptor-α; Estrogen receptor-β; GPER
R,R-THC
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Targets
Estrogen receptor-α; Estrogen receptor-β
raloxifene
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Targets
Estrogen receptor-α; Estrogen receptor-β; GPER; aldehyde oxidase 1
HPTE
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Targets
Estrogen receptor-β
tamoxifen
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Targets
CYP3A4; Estrogen receptor-α; Estrogen receptor-β; GPER; Maxi Cl-; VRAC
PHTPP
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Targets
Estrogen receptor-β
ospemifene
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Targets
Estrogen receptor-α; Estrogen receptor-β

Please note that chemical structures may not be available for all antagonists at this target. For more details please email us.

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