(-)-pentazocine

Ligand id: 1606

Name: (-)-pentazocine

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Structure and Physico-chemical Properties

2D Structure
Calculated Physico-chemical Properties
Hydrogen bond acceptors 1
Hydrogen bond donors 1
Rotatable bonds 2
Topological polar surface area 23.47
Molecular weight 285.21
XLogP 4.09
No. Lipinski's rules broken 0

Molecular properties generated using the CDK

No information available.
Summary of Clinical Use
Pentazocine is used to treat moderate to severe pain. It is also used as part of surgical anesthesia.
Mechanism Of Action and Pharmacodynamic Effects
Evidence suggests that pentazocine antagonizes the opioid effects by competing for the same receptor sites.