Ligand id: 1136

Name: glucagon

Species: Human, Mouse, Rat

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Structure and Physico-chemical Properties

2D Structure

View interactive charts of activity data from ChEMBL and GtoPdb across species (New!)

Natural/Endogenous Targets
GLP-1 receptor
glucagon receptor
Selectivity at Human GPCRs
Key to terms and symbols Click column headers to sort
Target Type Action Affinity Units Concentration range (M) Reference
GLP-1 receptor Agonist Full agonist 6.9 – 7.0 pKi - 1
pKi 6.9 – 7.0 [1]
glucagon receptor Agonist Full agonist 9.0 pEC50 - 2
pEC50 9.0 [2]
Ligand mentioned in the following text fields