apelin receptor early endogenous ligand

Ligand id: 7930

Name: apelin receptor early endogenous ligand

Abbreviated name: ELA

Species: Human

View interactive charts of activity data from GtoPdb and ChEMBL (where available) across species

Bioactivity Comments
Alkaline phosphatase-conjugated APELA has been demonstrated to bind to the human apelin receptor by in vitro colourimetric assay [1].
Natural/Endogenous Targets
apelin receptor
Selectivity at GPCRs
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Target Sp. Type Action Affinity Units Concentration range (M) Reference
apelin receptor Hs Agonist Agonist 9.3 pKd - 2
pKd 9.3 (Kd 5.1x10-10 M) [2]