ketanserin

Ligand id: 88

Name: ketanserin

Structure and Physico-chemical Properties

2D Structure
Calculated Physico-chemical Properties
Hydrogen bond acceptors 6
Hydrogen bond donors 1
Rotatable bonds 5
Topological polar surface area 69.72
Molecular weight 395.16
XLogP 3.33
No. Lipinski's rules broken 0

Molecular properties generated using the CDK

No information available.
Summary of Clinical Use
May be used as an anti-hypertensive. There is no information regarding approval for clinical use of this drug on the US FDA or European Medicines Agency websites. Individual national approval agencies may have granted marketing authorisation. The drug may also be approved for veterinary use.
Mechanism Of Action and Pharmacodynamic Effects
This drug has affinity for multiple GPCRs, including 5-HT2A, 5-HT2C5-HT2C, histamine H1, and α1-adrenoceptors.