Available chemical structures for AXL receptor tyrosine kinase inhibitors

canlitinib
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Targets
AXL receptor tyrosine kinase; kinase insert domain receptor
gilteritinib
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Targets
ALK receptor tyrosine kinase; AXL receptor tyrosine kinase; MER proto-oncogene, tyrosine kinase; c-ros oncogene 1, receptor tyrosine kinase; fms related receptor tyrosine kinase 3; leukocyte receptor tyrosine kinase; neurotrophic receptor tyrosine kinase 1; ret proto-oncogene
BMS-777607
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Targets
AXL receptor tyrosine kinase; MER proto-oncogene, tyrosine kinase; MET proto-oncogene, receptor tyrosine kinase; TYRO3 protein tyrosine kinase; macrophage stimulating 1 receptor
sitravatinib
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Targets
AXL receptor tyrosine kinase; EPH receptor A3; KIT proto-oncogene, receptor tyrosine kinase; MER proto-oncogene, tyrosine kinase; MET proto-oncogene, receptor tyrosine kinase; discoidin domain receptor tyrosine kinase 2; fms related receptor tyrosine kinase 1; fms related receptor tyrosine kinase 3; fms related receptor tyrosine kinase 4; kinase insert domain receptor; neurotrophic receptor tyrosine kinase 1; platelet derived growth factor receptor alpha
compound 6li [Chan et al., 2022]
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Targets
AXL receptor tyrosine kinase; KIT proto-oncogene, receptor tyrosine kinase; fms related receptor tyrosine kinase 3; tyrosine kinase with immunoglobulin like and EGF like domains 1
compound 8i [PMID: 22765894]
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Targets
AXL receptor tyrosine kinase; KIT proto-oncogene, receptor tyrosine kinase; MET proto-oncogene, receptor tyrosine kinase; TEK receptor tyrosine kinase; fibroblast growth factor receptor 1; fms related receptor tyrosine kinase 1; fms related receptor tyrosine kinase 3; fms related receptor tyrosine kinase 4; kinase insert domain receptor; macrophage stimulating 1 receptor; platelet derived growth factor receptor alpha; platelet derived growth factor receptor beta
UNC8969
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Targets
AXL receptor tyrosine kinase; MER proto-oncogene, tyrosine kinase; TYRO3 protein tyrosine kinase; fms related receptor tyrosine kinase 3
A-910
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Targets
AXL receptor tyrosine kinase; MER proto-oncogene, tyrosine kinase; TYRO3 protein tyrosine kinase
zanzalintinib
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Targets
AXL receptor tyrosine kinase; MER proto-oncogene, tyrosine kinase; MET proto-oncogene, receptor tyrosine kinase
merestinib
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Targets
AXL receptor tyrosine kinase; MER proto-oncogene, tyrosine kinase; MET proto-oncogene, receptor tyrosine kinase; TEK receptor tyrosine kinase; discoidin domain receptor tyrosine kinase 1; fms related receptor tyrosine kinase 3; macrophage stimulating 1 receptor; tyrosine kinase with immunoglobulin like and EGF like domains 1
ningetinib
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Targets
AXL receptor tyrosine kinase; MET proto-oncogene, receptor tyrosine kinase; kinase insert domain receptor
bemcentinib
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Targets
AXL receptor tyrosine kinase
dubermatinib
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Targets
AXL receptor tyrosine kinase; aurora kinase A; aurora kinase B
LDC1267
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Targets
AXL receptor tyrosine kinase; MER proto-oncogene, tyrosine kinase; TYRO3 protein tyrosine kinase
RIPK1 inhibitor 22b
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Targets
AXL receptor tyrosine kinase; MER proto-oncogene, tyrosine kinase; discoidin domain receptor tyrosine kinase 1; eukaryotic translation initiation factor 2 alpha kinase 1; fms related receptor tyrosine kinase 4; mitogen-activated protein kinase kinase kinase kinase 5; neurotrophic receptor tyrosine kinase 1; neurotrophic receptor tyrosine kinase 2; neurotrophic receptor tyrosine kinase 3; receptor interacting serine/threonine kinase 1; receptor interacting serine/threonine kinase 3
compound 19a [PMID: 30503936]
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Targets
AXL receptor tyrosine kinase; Insulin-like growth factor I receptor; KIT proto-oncogene, receptor tyrosine kinase; MET proto-oncogene, receptor tyrosine kinase; SRC proto-oncogene, non-receptor tyrosine kinase; epidermal growth factor receptor; kinase insert domain receptor; macrophage stimulating 1 receptor
SLC-391
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Targets
AXL receptor tyrosine kinase; MER proto-oncogene, tyrosine kinase; TYRO3 protein tyrosine kinase
compound 1 [Cruz-López et al., 2019]
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Targets
AXL receptor tyrosine kinase; fms related receptor tyrosine kinase 3
belizatinib
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Targets
ALK receptor tyrosine kinase; AXL receptor tyrosine kinase; LCK proto-oncogene, Src family tyrosine kinase; MER proto-oncogene, tyrosine kinase; fms related receptor tyrosine kinase 3; interleukin 1 receptor associated kinase 1; leukocyte receptor tyrosine kinase; mitogen-activated protein kinase kinase kinase kinase 2
adrixetinib
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Targets
AXL receptor tyrosine kinase; MER proto-oncogene, tyrosine kinase; colony stimulating factor 1 receptor
UNC4203
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Targets
AXL receptor tyrosine kinase; MER proto-oncogene, tyrosine kinase; TYRO3 protein tyrosine kinase; fms related receptor tyrosine kinase 3

Please note that chemical structures may not be available for all inhibitors at this target. For more details please email us.