Available chemical structures for Pim-1 proto-oncogene, serine/threonine kinase inhibitors

uzansertib
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Targets
Pim-1 proto-oncogene, serine/threonine kinase; Pim-2 proto-oncogene, serine/threonine kinase; Pim-3 proto-oncogene, serine/threonine kinase
leucettine L41
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Targets
CDC like kinase 1; CDC like kinase 3; Pim-1 proto-oncogene, serine/threonine kinase; dual specificity tyrosine phosphorylation regulated kinase 1A; dual specificity tyrosine phosphorylation regulated kinase 2; dual specificity tyrosine phosphorylation regulated kinase 4
compound 14k [PMID: 21982499]
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Targets
Pim-1 proto-oncogene, serine/threonine kinase; Pim-2 proto-oncogene, serine/threonine kinase; Pim-3 proto-oncogene, serine/threonine kinase; casein kinase 1 gamma 3; fms related receptor tyrosine kinase 3
CX-6258
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Targets
Pim-1 proto-oncogene, serine/threonine kinase; Pim-2 proto-oncogene, serine/threonine kinase; Pim-3 proto-oncogene, serine/threonine kinase
SGI-1776
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Targets
Pim-1 proto-oncogene, serine/threonine kinase; Pim-2 proto-oncogene, serine/threonine kinase; Pim-3 proto-oncogene, serine/threonine kinase; fms related receptor tyrosine kinase 3; histone H3 associated protein kinase
XL413
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Targets
Casein kinase 2; Pim-1 proto-oncogene, serine/threonine kinase; cell division cycle 7
compound 28 [PMID: 30624936]
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Targets
Pim-1 proto-oncogene, serine/threonine kinase; Pim-2 proto-oncogene, serine/threonine kinase
compound 20 [PMID: 22136433]
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Targets
Calmodulin-dependent kinase II; Pim-1 proto-oncogene, serine/threonine kinase; Pim-3 proto-oncogene, serine/threonine kinase; protein kinase N1
voruciclib
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Targets
LIM domain kinase 1; Pim-1 proto-oncogene, serine/threonine kinase; casein kinase 1 gamma 1; cyclin dependent kinase 1; cyclin dependent kinase 2; cyclin dependent kinase 4; cyclin dependent kinase 5; cyclin dependent kinase 6; cyclin dependent kinase 8; cyclin dependent kinase 9; dual specificity tyrosine phosphorylation regulated kinase 1B; glycogen synthase kinase 3 alpha; glycogen synthase kinase 3 beta; mitogen-activated protein kinase kinase 2
ruboxistaurin
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Targets
Pim-1 proto-oncogene, serine/threonine kinase; Pim-2 proto-oncogene, serine/threonine kinase; protein kinase C alpha; protein kinase C beta; protein kinase C delta; protein kinase C gamma
silmitasertib
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Targets
Pim-1 proto-oncogene, serine/threonine kinase; casein kinase 2, alpha 1 polypeptide subunit; casein kinase 2, alpha prime polypeptide subunit; death associated protein kinase 3; homeodomain interacting protein kinase 3
compound 2 [PMID: 22560567]
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Targets
CDC like kinase 1; Casein kinase 2; Pim-1 proto-oncogene, serine/threonine kinase; cell division cycle 7; glycogen synthase kinase 3 beta
Akt inhibitor X
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Targets
Pim-1 proto-oncogene, serine/threonine kinase
CX-5011
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Targets
Casein kinase 2; Pim-1 proto-oncogene, serine/threonine kinase
CX-5279
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Targets
Casein kinase 2; Pim-1 proto-oncogene, serine/threonine kinase
LGB321
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Targets
Pim-1 proto-oncogene, serine/threonine kinase; Pim-2 proto-oncogene, serine/threonine kinase; Pim-3 proto-oncogene, serine/threonine kinase
PIM447
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Targets
Pim-1 proto-oncogene, serine/threonine kinase; Pim-2 proto-oncogene, serine/threonine kinase; Pim-3 proto-oncogene, serine/threonine kinase
AZD1208
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Targets
Pim-1 proto-oncogene, serine/threonine kinase; Pim-2 proto-oncogene, serine/threonine kinase; Pim-3 proto-oncogene, serine/threonine kinase
GDC-0339
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Targets
Pim-1 proto-oncogene, serine/threonine kinase; Pim-2 proto-oncogene, serine/threonine kinase; Pim-3 proto-oncogene, serine/threonine kinase
nuvisertib
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Targets
Pim-1 proto-oncogene, serine/threonine kinase; Pim-2 proto-oncogene, serine/threonine kinase; Pim-3 proto-oncogene, serine/threonine kinase; fms related receptor tyrosine kinase 3
dapolsertib
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Targets
Pim-1 proto-oncogene, serine/threonine kinase; Pim-2 proto-oncogene, serine/threonine kinase; Pim-3 proto-oncogene, serine/threonine kinase

Please note that chemical structures may not be available for all inhibitors at this target. For more details please email us.