Available chemical structures for fibroblast growth factor receptor 3 inhibitors

futibatinib
Click here for ligand page
Targets
fibroblast growth factor receptor 1; fibroblast growth factor receptor 2; fibroblast growth factor receptor 3; fibroblast growth factor receptor 4
infigratinib
Click here for ligand page
Targets
fibroblast growth factor receptor 1; fibroblast growth factor receptor 2; fibroblast growth factor receptor 3; fibroblast growth factor receptor 4; kinase insert domain receptor
compound 29 [PMID: 36356320]
Click here for ligand page
Targets
fibroblast growth factor receptor 1; fibroblast growth factor receptor 2; fibroblast growth factor receptor 3; fibroblast growth factor receptor 4
ASP5878
Click here for ligand page
Targets
fibroblast growth factor receptor 3
erdafitinib
Click here for ligand page
Targets
fibroblast growth factor receptor 1; fibroblast growth factor receptor 2; fibroblast growth factor receptor 3; fibroblast growth factor receptor 4; kinase insert domain receptor
tinengotinib
Click here for ligand page
Targets
Janus kinase 2; aurora kinase A; aurora kinase B; fibroblast growth factor receptor 1; fibroblast growth factor receptor 3; fms related receptor tyrosine kinase 1; kinase insert domain receptor
segigratinib
Click here for ligand page
Targets
colony stimulating factor 1 receptor; fibroblast growth factor receptor 1; fibroblast growth factor receptor 2; fibroblast growth factor receptor 3; fibroblast growth factor receptor 4
PRN1371
Click here for ligand page
Targets
fibroblast growth factor receptor 1; fibroblast growth factor receptor 2; fibroblast growth factor receptor 3; fibroblast growth factor receptor 4
derazantinib
Click here for ligand page
Targets
fibroblast growth factor receptor 1; fibroblast growth factor receptor 2; fibroblast growth factor receptor 3
fexagratinib
Click here for ligand page
Targets
Insulin-like growth factor I receptor; fibroblast growth factor receptor 1; fibroblast growth factor receptor 2; fibroblast growth factor receptor 3; fibroblast growth factor receptor 4; kinase insert domain receptor
dovitinib
Click here for ligand page
Targets
Insulin receptor; KIT proto-oncogene, receptor tyrosine kinase; colony stimulating factor 1 receptor; epidermal growth factor receptor; fibroblast growth factor receptor 1; fibroblast growth factor receptor 3; fms related receptor tyrosine kinase 1; fms related receptor tyrosine kinase 3; fms related receptor tyrosine kinase 4; kinase insert domain receptor; platelet derived growth factor receptor alpha; platelet derived growth factor receptor beta
tasurgratinib
Click here for ligand page
Targets
fibroblast growth factor receptor 1; fibroblast growth factor receptor 2; fibroblast growth factor receptor 3; fibroblast growth factor receptor 4
compound 7 [Nguyen et al., 2023]
Click here for ligand page
Targets
activin A receptor type 1; fibroblast growth factor receptor 1; fibroblast growth factor receptor 2; fibroblast growth factor receptor 3; fibroblast growth factor receptor 4
fanregratinib
Click here for ligand page
Targets
fibroblast growth factor receptor 1; fibroblast growth factor receptor 2; fibroblast growth factor receptor 3
LY2874455
Click here for ligand page
Targets
fibroblast growth factor receptor 1; fibroblast growth factor receptor 2; fibroblast growth factor receptor 3; fibroblast growth factor receptor 4; kinase insert domain receptor
dabogratinib
Click here for ligand page
Targets
fibroblast growth factor receptor 1; fibroblast growth factor receptor 2; fibroblast growth factor receptor 3; fibroblast growth factor receptor 4
zoligratinib
Click here for ligand page
Targets
fibroblast growth factor receptor 1; fibroblast growth factor receptor 2; fibroblast growth factor receptor 3; fibroblast growth factor receptor 4; platelet derived growth factor receptor beta
rogaratinib
Click here for ligand page
Targets
fibroblast growth factor receptor 1; fibroblast growth factor receptor 3
MK-2461
Click here for ligand page
Targets
MER proto-oncogene, tyrosine kinase; MET proto-oncogene, receptor tyrosine kinase; fibroblast growth factor receptor 1; fibroblast growth factor receptor 2; fibroblast growth factor receptor 3; fms related receptor tyrosine kinase 1; fms related receptor tyrosine kinase 3; fms related receptor tyrosine kinase 4; kinase insert domain receptor; macrophage stimulating 1 receptor; neurotrophic receptor tyrosine kinase 1; neurotrophic receptor tyrosine kinase 2; platelet derived growth factor receptor beta
pemigatinib
Click here for ligand page
Targets
fibroblast growth factor receptor 1; fibroblast growth factor receptor 2; fibroblast growth factor receptor 3
nintedanib
Click here for ligand page
Targets
fibroblast growth factor receptor 1; fibroblast growth factor receptor 2; fibroblast growth factor receptor 3; fibroblast growth factor receptor 4; fms related receptor tyrosine kinase 1; fms related receptor tyrosine kinase 4; kinase insert domain receptor; large tumor suppressor kinase 1; platelet derived growth factor receptor alpha; platelet derived growth factor receptor beta
compound 1d [PMID: 21493067]
Click here for ligand page
Targets
Janus kinase 2; Janus kinase 3; fibroblast growth factor receptor 3; muscle associated receptor tyrosine kinase; neurotrophic receptor tyrosine kinase 1; ret proto-oncogene
BLU-9931
Click here for ligand page
Targets
fibroblast growth factor receptor 1; fibroblast growth factor receptor 2; fibroblast growth factor receptor 3; fibroblast growth factor receptor 4
TAK-632
Click here for ligand page
Targets
B-Raf proto-oncogene, serine/threonine kinase; Raf-1 proto-oncogene, serine/threonine kinase; aurora kinase B; fibroblast growth factor receptor 3; platelet derived growth factor receptor beta; receptor interacting serine/threonine kinase 1; receptor interacting serine/threonine kinase 3

Please note that chemical structures may not be available for all inhibitors at this target. For more details please email us.