Available chemical structures for LPA1 receptor antagonists

AM966
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Targets
LPA1 receptor; LPA2 receptor; LPA3 receptor; LPA4 receptor
BMS-986020
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Targets
LPA1 receptor
ACT-1016-0707
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Targets
LPA1 receptor
ONO-3080573
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Targets
LPA1 receptor
ONO-9910539
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Targets
LPA1 receptor
ONO-9780307
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Targets
LPA1 receptor
mianserin
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Targets
α1A-adrenoceptor; α1B-adrenoceptor; α1D-adrenoceptor; 5-HT1B receptor; 5-HT2A receptor; 5-HT2B receptor; 5-HT2C receptor; 5-HT6 receptor; 5-HT7 receptor; NET
SAR100842
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Targets
LPA1 receptor
VPC32183
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Targets
LPA1 receptor; LPA3 receptor
ONO-7300243
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Targets
LPA1 receptor
Ki16425
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Targets
GPR87; LPA1 receptor; LPA2 receptor; LPA3 receptor
amitriptyline
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Targets
α1A-adrenoceptor; 5-HT2A receptor; 5-HT2C receptor; 5-HT6 receptor; 5-HT7 receptor; H1 receptor; M1 receptor; M2 receptor; M3 receptor; M4 receptor; M5 receptor; NET; SERT
syn-BrP-LPA
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Targets
LPA1 receptor
AM095
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Targets
LPA1 receptor
anti-BrP-LPA
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Targets
LPA1 receptor
BrP-LPA
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Targets
LPA1 receptor; LPA2 receptor
BMS-986278
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Targets
LPA1 receptor
VPC12249
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Targets
LPA1 receptor; LPA3 receptor; S1P3 receptor
dioctanoylglycerol pyrophosphate
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Targets
GPR87; P2RY10; LPA1 receptor; LPA3 receptor
VPC32179
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Targets
LPA1 receptor; LPA3 receptor

Please note that chemical structures may not be available for all antagonists at this target. For more details please email us.

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