Available chemical structures for platelet derived growth factor receptor beta inhibitors

CP-673451
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Targets
KIT proto-oncogene, receptor tyrosine kinase; platelet derived growth factor receptor alpha; platelet derived growth factor receptor beta
compound 8h [PMID: 22765894]
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Targets
KIT proto-oncogene, receptor tyrosine kinase; SRC proto-oncogene, non-receptor tyrosine kinase; fibroblast growth factor receptor 1; fms related receptor tyrosine kinase 1; fms related receptor tyrosine kinase 3; fms related receptor tyrosine kinase 4; kinase insert domain receptor; mitogen-activated protein kinase kinase kinase kinase 3; platelet derived growth factor receptor alpha; platelet derived growth factor receptor beta; ribosomal protein S6 kinase A3
compound 8i [PMID: 22765894]
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Targets
AXL receptor tyrosine kinase; KIT proto-oncogene, receptor tyrosine kinase; MET proto-oncogene, receptor tyrosine kinase; TEK receptor tyrosine kinase; fibroblast growth factor receptor 1; fms related receptor tyrosine kinase 1; fms related receptor tyrosine kinase 3; fms related receptor tyrosine kinase 4; kinase insert domain receptor; macrophage stimulating 1 receptor; platelet derived growth factor receptor alpha; platelet derived growth factor receptor beta
M4205
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Targets
KIT proto-oncogene, receptor tyrosine kinase; colony stimulating factor 1 receptor; platelet derived growth factor receptor alpha; platelet derived growth factor receptor beta
SU11652
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Targets
KIT proto-oncogene, receptor tyrosine kinase; fibroblast growth factor receptor 1; kinase insert domain receptor; platelet derived growth factor receptor beta
SU-14813
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Targets
KIT proto-oncogene, receptor tyrosine kinase; fibroblast growth factor receptor 1; fms related receptor tyrosine kinase 1; kinase insert domain receptor; platelet derived growth factor receptor beta
famitinib
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Targets
KIT proto-oncogene, receptor tyrosine kinase; kinase insert domain receptor; platelet derived growth factor receptor beta
PDGF receptor tyrosine kinase inhibitor IV
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Targets
platelet derived growth factor receptor beta
cediranib
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Targets
KIT proto-oncogene, receptor tyrosine kinase; colony stimulating factor 1 receptor; fms related receptor tyrosine kinase 1; fms related receptor tyrosine kinase 3; fms related receptor tyrosine kinase 4; kinase insert domain receptor; platelet derived growth factor receptor alpha; platelet derived growth factor receptor beta
sunitinib
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Targets
KIT proto-oncogene, receptor tyrosine kinase; fibroblast growth factor receptor 1; fms related receptor tyrosine kinase 3; fms related receptor tyrosine kinase 4; kinase insert domain receptor; large tumor suppressor kinase 1; large tumor suppressor kinase 2; platelet derived growth factor receptor beta; ret proto-oncogene
lucitanib
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Targets
KIT proto-oncogene, receptor tyrosine kinase; fibroblast growth factor receptor 1; fms related receptor tyrosine kinase 1; kinase insert domain receptor; platelet derived growth factor receptor alpha; platelet derived growth factor receptor beta; ret proto-oncogene
henatinib
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Targets
KIT proto-oncogene, receptor tyrosine kinase; kinase insert domain receptor; platelet derived growth factor receptor beta
dovitinib
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Targets
Insulin receptor; KIT proto-oncogene, receptor tyrosine kinase; colony stimulating factor 1 receptor; epidermal growth factor receptor; fibroblast growth factor receptor 1; fibroblast growth factor receptor 3; fms related receptor tyrosine kinase 1; fms related receptor tyrosine kinase 3; fms related receptor tyrosine kinase 4; kinase insert domain receptor; platelet derived growth factor receptor alpha; platelet derived growth factor receptor beta
PDGF RTK inhibitor
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Targets
platelet derived growth factor receptor beta
ilorasertib
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Targets
KIT proto-oncogene, receptor tyrosine kinase; aurora kinase A; aurora kinase B; aurora kinase C; colony stimulating factor 1 receptor; fms related receptor tyrosine kinase 1; fms related receptor tyrosine kinase 3; fms related receptor tyrosine kinase 4; kinase insert domain receptor; platelet derived growth factor receptor alpha; platelet derived growth factor receptor beta
tafetinib
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Targets
fms related receptor tyrosine kinase 3; fms related receptor tyrosine kinase 4; kinase insert domain receptor; platelet derived growth factor receptor beta; ret proto-oncogene
MK-2461
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Targets
MER proto-oncogene, tyrosine kinase; MET proto-oncogene, receptor tyrosine kinase; fibroblast growth factor receptor 1; fibroblast growth factor receptor 2; fibroblast growth factor receptor 3; fms related receptor tyrosine kinase 1; fms related receptor tyrosine kinase 3; fms related receptor tyrosine kinase 4; kinase insert domain receptor; macrophage stimulating 1 receptor; neurotrophic receptor tyrosine kinase 1; neurotrophic receptor tyrosine kinase 2; platelet derived growth factor receptor beta
KBP-7018
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Targets
KIT proto-oncogene, receptor tyrosine kinase; platelet derived growth factor receptor beta; ret proto-oncogene
BPR1R024
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Targets
KIT proto-oncogene, receptor tyrosine kinase; colony stimulating factor 1 receptor; platelet derived growth factor receptor alpha; platelet derived growth factor receptor beta
orantinib
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Targets
epidermal growth factor receptor; fibroblast growth factor receptor 1; kinase insert domain receptor; platelet derived growth factor receptor beta
sorafenib
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Targets
B-Raf proto-oncogene, serine/threonine kinase; KIT proto-oncogene, receptor tyrosine kinase; Raf-1 proto-oncogene, serine/threonine kinase; TNNI3 interacting kinase; cyclin dependent kinase 19; cyclin dependent kinase 8; discoidin domain receptor tyrosine kinase 2; fibroblast growth factor receptor 1; fms related receptor tyrosine kinase 3; fms related receptor tyrosine kinase 4; kinase insert domain receptor; platelet derived growth factor receptor beta; ret proto-oncogene
nintedanib
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Targets
fibroblast growth factor receptor 1; fibroblast growth factor receptor 2; fibroblast growth factor receptor 3; fibroblast growth factor receptor 4; fms related receptor tyrosine kinase 1; fms related receptor tyrosine kinase 4; kinase insert domain receptor; large tumor suppressor kinase 1; platelet derived growth factor receptor alpha; platelet derived growth factor receptor beta
linifanib
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Targets
KIT proto-oncogene, receptor tyrosine kinase; TEK receptor tyrosine kinase; colony stimulating factor 1 receptor; cyclin dependent kinase 19; cyclin dependent kinase 8; fms related receptor tyrosine kinase 1; fms related receptor tyrosine kinase 3; fms related receptor tyrosine kinase 4; kinase insert domain receptor; platelet derived growth factor receptor beta; ret proto-oncogene
PDGF receptor tyrosine kinase inhibitor III
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Targets
platelet derived growth factor receptor beta
pazopanib
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Targets
KIT proto-oncogene, receptor tyrosine kinase; colony stimulating factor 1 receptor; fibroblast growth factor receptor 1; fms related receptor tyrosine kinase 1; fms related receptor tyrosine kinase 4; kinase insert domain receptor; platelet derived growth factor receptor beta
AGL 2043
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Targets
platelet derived growth factor receptor beta
ibcasertib
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Targets
KIT proto-oncogene, receptor tyrosine kinase; aurora kinase B; colony stimulating factor 1 receptor; fms related receptor tyrosine kinase 1; fms related receptor tyrosine kinase 4; kinase insert domain receptor; platelet derived growth factor receptor alpha; platelet derived growth factor receptor beta
CHMFL-KIT-64
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Targets
KIT proto-oncogene, receptor tyrosine kinase; colony stimulating factor 1 receptor; discoidin domain receptor tyrosine kinase 1; fms related receptor tyrosine kinase 4; platelet derived growth factor receptor alpha; platelet derived growth factor receptor beta
TAK-632
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Targets
B-Raf proto-oncogene, serine/threonine kinase; Raf-1 proto-oncogene, serine/threonine kinase; aurora kinase B; fibroblast growth factor receptor 3; platelet derived growth factor receptor beta; receptor interacting serine/threonine kinase 1; receptor interacting serine/threonine kinase 3
Flt-3 inhibitor II
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Targets
fms related receptor tyrosine kinase 3; platelet derived growth factor receptor beta
tandutinib
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Targets
KIT proto-oncogene, receptor tyrosine kinase; colony stimulating factor 1 receptor; fms related receptor tyrosine kinase 3; platelet derived growth factor receptor beta
Ki-20227
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Targets
KIT proto-oncogene, receptor tyrosine kinase; colony stimulating factor 1 receptor; kinase insert domain receptor; platelet derived growth factor receptor beta
flumbatinib
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Targets
ABL proto-oncogene 1, non-receptor tyrosine kinase; KIT proto-oncogene, receptor tyrosine kinase; platelet derived growth factor receptor beta
SU5402
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Targets
fibroblast growth factor receptor 1; kinase insert domain receptor; platelet derived growth factor receptor beta
zoligratinib
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Targets
fibroblast growth factor receptor 1; fibroblast growth factor receptor 2; fibroblast growth factor receptor 3; fibroblast growth factor receptor 4; platelet derived growth factor receptor beta
vatalanib
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Targets
fms related receptor tyrosine kinase 1; fms related receptor tyrosine kinase 4; kinase insert domain receptor; platelet derived growth factor receptor beta
semaxanib
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Targets
KIT proto-oncogene, receptor tyrosine kinase; fms related receptor tyrosine kinase 1; kinase insert domain receptor; platelet derived growth factor receptor beta
masitinib
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Targets
KIT proto-oncogene, receptor tyrosine kinase; platelet derived growth factor receptor alpha; platelet derived growth factor receptor beta
GTP-14564
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Targets
KIT proto-oncogene, receptor tyrosine kinase; colony stimulating factor 1 receptor; fms related receptor tyrosine kinase 3; platelet derived growth factor receptor beta
sotuletinib
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Targets
KIT proto-oncogene, receptor tyrosine kinase; colony stimulating factor 1 receptor; platelet derived growth factor receptor beta
AC710
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Targets
KIT proto-oncogene, receptor tyrosine kinase; colony stimulating factor 1 receptor; fms related receptor tyrosine kinase 3; platelet derived growth factor receptor alpha; platelet derived growth factor receptor beta
crenolanib
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Targets
KIT proto-oncogene, receptor tyrosine kinase; colony stimulating factor 1 receptor; fms related receptor tyrosine kinase 3; platelet derived growth factor receptor alpha; platelet derived growth factor receptor beta
quizartinib
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Targets
KIT proto-oncogene, receptor tyrosine kinase; colony stimulating factor 1 receptor; fms related receptor tyrosine kinase 3; platelet derived growth factor receptor alpha; platelet derived growth factor receptor beta; ret proto-oncogene
naporafenib
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Targets
B-Raf proto-oncogene, serine/threonine kinase; Raf-1 proto-oncogene, serine/threonine kinase; discoidin domain receptor tyrosine kinase 1; discoidin domain receptor tyrosine kinase 2; platelet derived growth factor receptor beta
compound 5e [PMID: 28580438]
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Targets
Janus kinase 1; fms related receptor tyrosine kinase 3; platelet derived growth factor receptor beta
IACS-9439
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Targets
colony stimulating factor 1 receptor; platelet derived growth factor receptor beta
salvianolic acid B
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Targets
CD226 molecule; lysine demethylase 1A; platelet derived growth factor receptor beta
PD166285
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Targets
SRC proto-oncogene, non-receptor tyrosine kinase; WEE1 G2 checkpoint kinase; epidermal growth factor receptor; fibroblast growth factor receptor 1; platelet derived growth factor receptor beta; protein kinase, membrane associated tyrosine/threonine 1
seralutinib
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Targets
platelet derived growth factor receptor alpha; platelet derived growth factor receptor beta

Please note that chemical structures may not be available for all inhibitors at this target. For more details please email us.