PF‐06928215 [Ligand Id: 11324] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Cyclic GMP-AMP synthase in Human [GtoPdb: 3165] [UniProtKB: Q8N884] | ||||||||
| GtoPdb | Binding affinity determined by SPR. | - | 6.7 | pKd | 200 | nM | Kd | PLoS One (2017) 12: e0184843 [PMID:28934246] |
| GtoPdb | Enzyme inhibition determined by FP assay. | - | 5.31 | pIC50 | 4900 | nM | IC50 | PLoS One (2017) 12: e0184843 [PMID:28934246] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
