nacresertib [Ligand Id: 13502] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| interleukin 1 receptor associated kinase 1 in Human [GtoPdb: 2042] [UniProtKB: P51617] | ||||||||
| GtoPdb | - | - | 5.39 | pIC50 | 4039 | nM | IC50 | WO2021057785A1. Irak inhibitor and preparation method therefor and use thereof (2021) |
| interleukin 1 receptor associated kinase 4 in Human [GtoPdb: 2045] [UniProtKB: Q9NWZ3] | ||||||||
| GtoPdb | Measuring inhibtion of IRAK4-mediated substrate phosphorylation in a mobility-shift assay | - | 8.22 | pIC50 | 6 | nM | IC50 | WO2021057785A1. Irak inhibitor and preparation method therefor and use thereof (2021) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
