setanaxib [Ligand Id: 9932] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • NADPH oxidase 1 in Human [GtoPdb: 3001] [UniProtKB: Q9Y5S8]
There should be some charts here, you may need to enable JavaScript!
  • cytochrome b-245 beta chain in Human [GtoPdb: 3002] [UniProtKB: P04839]
There should be some charts here, you may need to enable JavaScript!
  • NADPH oxidase 4 in Human [GtoPdb: 3004] [UniProtKB: Q9NPH5]
There should be some charts here, you may need to enable JavaScript!
  • NADPH oxidase 5 in Human [GtoPdb: 3005] [UniProtKB: Q96PH1]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
NADPH oxidase 1 in Human [GtoPdb: 3001] [UniProtKB: Q9Y5S8]
GtoPdb - - 6.85 pKi 140 nM Ki Hepatology (2012) 56: 2316-27 [PMID:22806357]
cytochrome b-245 beta chain in Human [GtoPdb: 3002] [UniProtKB: P04839]
GtoPdb - - 5.76 pKi 1750 nM Ki Hepatology (2012) 56: 2316-27 [PMID:22806357]
NADPH oxidase 4 in Human [GtoPdb: 3004] [UniProtKB: Q9NPH5]
GtoPdb - - 6.96 pKi 110 nM Ki Hepatology (2012) 56: 2316-27 [PMID:22806357]
NADPH oxidase 5 in Human [GtoPdb: 3005] [UniProtKB: Q96PH1]
GtoPdb - - 6.39 pKi 410 nM Ki Hepatology (2012) 56: 2316-27 [PMID:22806357]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.