triple modulator 10 [PMID: 29878767] [Ligand Id: 10002] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| CysLT1 receptor in Human [GtoPdb: 269] [UniProtKB: Q9Y271] | ||||||||
| GtoPdb | - | - | 8.7 | pA2 | - | - | - | J Med Chem (2018) 61: 5758-5764 [PMID:29878767] |
| Peroxisome proliferator-activated receptor-γ in Human [GtoPdb: 595] [UniProtKB: P37231] | ||||||||
| GtoPdb | - | - | 6.52 | pEC50 | 300 | nM | EC50 | J Med Chem (2018) 61: 5758-5764 [PMID:29878767] |
| epoxide hydrolase 2 in Human [GtoPdb: 2970] [UniProtKB: P34913] | ||||||||
| GtoPdb | - | - | 7.37 | pIC50 | 43 | nM | IC50 | J Med Chem (2018) 61: 5758-5764 [PMID:29878767] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
