cintirorgon [Ligand Id: 10045] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| RAR-related orphan receptor-γ in Human [GtoPdb: 600] [UniProtKB: P51449] | ||||||||
| GtoPdb | Measured in a RORγ-ligand binding domain TR-FRET assay. | - | 6.3 | pEC50 | <500 | nM | EC50 | WO2016201225A1. Aryl dihydro-2h-benzo[b][1,4]oxazine sulfonamide and related compounds for use as agonists of rory and the treatment of disease (2016) |
| GtoPdb | Measured in a RORγ-ligand binding domain Gal4-RORγ luciferase reporter assay. | - | 6.3 | pEC50 | <500 | nM | EC50 | WO2016201225A1. Aryl dihydro-2h-benzo[b][1,4]oxazine sulfonamide and related compounds for use as agonists of rory and the treatment of disease (2016) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
