compound 3f [Festa et al., 2019] [Ligand Id: 10187] activity data from GtoPdb

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  • Farnesoid X receptor in Human [GtoPdb: 603] [UniProtKB: Q96RI1]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Farnesoid X receptor in Human [GtoPdb: 603] [UniProtKB: Q96RI1]
GtoPdb Cellular potency (HepG2 cells) measured as antagonism of CDCA-induced FXR activation in a transactivation reporter assay. - 6.24 pIC50 580 nM IC50 ACS Med Chem Lett (2019) 10: 504-510 [PMID:30996787]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.