compound 28 [PMID: 30624936] [Ligand Id: 10195] activity data from GtoPdb

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  • Pim-1 proto-oncogene, serine/threonine kinase in Human [GtoPdb: 2158] [UniProtKB: P11309]
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  • Pim-2 proto-oncogene, serine/threonine kinase in Human [GtoPdb: 2159] [UniProtKB: Q9P1W9]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Pim-1 proto-oncogene, serine/threonine kinase in Human [GtoPdb: 2158] [UniProtKB: P11309]
GtoPdb - - 7.3 pIC50 50 nM IC50 J Med Chem (2019) 62: 1523-1540 [PMID:30624936]
Pim-2 proto-oncogene, serine/threonine kinase in Human [GtoPdb: 2159] [UniProtKB: Q9P1W9]
GtoPdb - - 7.3 pIC50 50 nM IC50 J Med Chem (2019) 62: 1523-1540 [PMID:30624936]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.