VU0810464 [Ligand Id: 10260] activity data from GtoPdb

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  • Kir3.1 in Human [GtoPdb: 434] [UniProtKB: P48549]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Kir3.1 in Human [GtoPdb: 434] [UniProtKB: P48549]
GtoPdb Activation of Kir3.1/3.4 (cardiac type) multimeric channels expressed in HEK-293 cells. - 6.14 pEC50 720 nM EC50 ACS Chem Neurosci (2017) 8: 1873-1879 [PMID:28697302]
GtoPdb Activation of Kir - 6.78 pEC50 165 nM EC50 ACS Chem Neurosci (2017) 8: 1873-1879 [PMID:28697302]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.