CIM0216 [Ligand Id: 10297] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • TRPM3 in Human [GtoPdb: 495] [UniProtKB: Q9HCF6]
  • TRPM3 in Mouse [GtoPdb: 495]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
TRPM3 in Human [GtoPdb: 495] [UniProtKB: Q9HCF6]
GtoPdb - - 6.1 pEC50 - - - Pharmacol Res (2017) 124: 92-99 [PMID:28720517];
Proc Natl Acad Sci USA (2015) 112: E1363-72 [PMID:25733887]
TRPM3 in Mouse [GtoPdb: 495]
GtoPdb Activation of outwardly rectifying currents in HEK293T cells expressing TRPM3α1 (long pore loop) variant - 6.12 pEC50 750 nM EC50 Br J Pharmacol (2022) 179: 3560-3575 [PMID:32780479]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.