selitrectinib [Ligand Id: 10314] activity data from GtoPdb
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| neurotrophic receptor tyrosine kinase 1 in Human [GtoPdb: 1817] [UniProtKB: P04629] | ||||||||
| GtoPdb | - | - | 9.3 | pIC50 | <0.5 | nM | IC50 | WO2017075107A1. Point mutations in trk inhibitor-resistant cancer and methods relating to the same (2017) |
| neurotrophic receptor tyrosine kinase 2 in Human [GtoPdb: 1818] [UniProtKB: Q16620] | ||||||||
| GtoPdb | - | - | 8.49 | pIC50 | 3.2 | nM | IC50 | WO2017075107A1. Point mutations in trk inhibitor-resistant cancer and methods relating to the same (2017) |
| neurotrophic receptor tyrosine kinase 3 in Human [GtoPdb: 1819] [UniProtKB: Q16288] | ||||||||
| GtoPdb | - | - | 8.6 | pIC50 | <2.5 | nM | IC50 | WO2017075107A1. Point mutations in trk inhibitor-resistant cancer and methods relating to the same (2017) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
