GS-444217 [Ligand Id: 10430] activity data from GtoPdb

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  • mitogen-activated protein kinase kinase kinase 5 in Human [GtoPdb: 2080] [UniProtKB: Q99683]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
mitogen-activated protein kinase kinase kinase 5 in Human [GtoPdb: 2080] [UniProtKB: Q99683]
GtoPdb Determined in a TR-FRET immunoassay. - 8.54 pIC50 2.9 nM IC50 Diabetes (2015) 64: 3903-13 [PMID:26180085]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.