elsubrutinib [Ligand Id: 10464] activity data from GtoPdb

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  • Bruton tyrosine kinase in Human [GtoPdb: 1948] [UniProtKB: Q06187]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Bruton tyrosine kinase in Human [GtoPdb: 1948] [UniProtKB: Q06187]
GtoPdb Inhibition of BTK catalytic domain as measured using TR-FRET based detection of phosphorylated peptide Biotin-(Ahx)-GAEEEIYAAFFA-COOH, - 7 pIC50 <100 nM IC50 WO2014210255A1. Primary carboxamides as BTK inhibitors (2014)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.