mitapivat [Ligand Id: 10473] activity data from GtoPdb

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  • pyruvate kinase M1/2 in Human [GtoPdb: 3006] [UniProtKB: P14618]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
pyruvate kinase M1/2 in Human [GtoPdb: 3006] [UniProtKB: P14618]
GtoPdb Activation of the PKM2 isoform. - 7 pEC50 <100 nM EC50 WO2011002817A1. Therapeutic compounds and compositions (2011)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.