compound 1 [PMID: 31477924] [Ligand Id: 10481] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • discoidin domain receptor tyrosine kinase 1 in Human [GtoPdb: 1843] [UniProtKB: Q08345]
There should be some charts here, you may need to enable JavaScript!
  • discoidin domain receptor tyrosine kinase 2 in Human [GtoPdb: 1844] [UniProtKB: Q16832]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
discoidin domain receptor tyrosine kinase 1 in Human [GtoPdb: 1843] [UniProtKB: Q08345]
GtoPdb In vitro inhibitory activity in an enzymatic kinase assay. - 8 pIC50 10 nM IC50 Nat Biotechnol (2019) 37: 1038-1040 [PMID:31477924]
discoidin domain receptor tyrosine kinase 2 in Human [GtoPdb: 1844] [UniProtKB: Q16832]
GtoPdb In vitro inhibitory activity in an enzymatic kinase assay. - 6.63 pIC50 234 nM IC50 Nat Biotechnol (2019) 37: 1038-1040 [PMID:31477924]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.