3β-OH [Ligand Id: 10537] activity data from GtoPdb

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  • Cav3.2 in Rat [GtoPdb: 536] [UniProtKB: Q9EQ60]
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  • Cav3.3 in Rat [GtoPdb: 537] [UniProtKB: Q9Z0Y8]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Cav3.2 in Rat [GtoPdb: 536] [UniProtKB: Q9EQ60]
GtoPdb Inhibition of currents via native Cav3.2 currents in rat dorsal root ganglion cells. - 5.52 pIC50 3000 nM IC50 Br J Anaesth (2018) 120: 768-778 [PMID:29576117]
Cav3.3 in Rat [GtoPdb: 537] [UniProtKB: Q9Z0Y8]
GtoPdb Inhibition of currents via native Cav3.3 currents in rat reticular thalamic nucleus. - 5.7 pIC50 2000 nM IC50 Br J Anaesth (2018) 120: 768-778 [PMID:29576117]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.