ChEMBL ligand: CHEMBL539 (Acetasol, Acetic, Acetic acid, Acetic Acid, Acetic acid, diluted, Acetic acid glacial, Acetic acid,glacial, Acetic acid, glacial, Acetic Acid, Glacial, Aceticum acidum, Acetopyrine, Acidum aceticum, Acidum aceticum glaciale, Aci-jel, Acopyrine, Antipyrine acetylsalicylate, Distilled vinegar, E260, E-260, Earcalm, FEMA NO. 2006, Glacial acetic acid, INS-260, INS NO.260, NSC-111201, NSC-112209, NSC-115870, NSC-127175, NSC-132953, NSC-406306, Orlex, Orthoacetic acid, Pyrosal, Vinegar, Vinegar acid, Vosol)
FFA3 receptor/Free fatty acid receptor 3 in Human [ChEMBL: CHEMBL5201] [GtoPdb: 227] [UniProtKB: O14843] There should be some charts here, you may need to enable JavaScript!
FYN proto-oncogene, Src family tyrosine kinase/Tyrosine-protein kinase FYN in Human [ChEMBL: CHEMBL1841] [GtoPdb: 2026] [UniProtKB: P06241] There should be some charts here, you may need to enable JavaScript!
LCK proto-oncogene, Src family tyrosine kinase/Tyrosine-protein kinase LCK in Human [ChEMBL: CHEMBL258] [GtoPdb: 2053] [UniProtKB: P06239] There should be some charts here, you may need to enable JavaScript!
FFA2 receptor in Human [GtoPdb: 226] [UniProtKB: O15552] There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
FFA3 receptor/Free fatty acid receptor 3 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL5201] [GtoPdb: 227] [UniProtKB: O14843]
GtoPdb	-	-	3.9	pEC50	-	-	-	J Biol Chem (2003) 278: 11312-9 [PMID:12496283]; J Biol Chem (2003) 278: 25481-9 [PMID:12711604]; Proc Natl Acad Sci USA (2004) 101: 1045-50 [PMID:14722361]; J Biol Chem (2011) 286: 10628-40 [PMID:21220428]
ChEMBL	Agonist activity at human GPCR41 transfected in HEK293 cells assessed as [35S]GTPgammaS binding by scintillation counting method	F	4.92	pEC50	12000	nM	EC50	J Med Chem (2018) 61: 47-61 [PMID:28745893]
FYN proto-oncogene, Src family tyrosine kinase/Tyrosine-protein kinase FYN in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1841] [GtoPdb: 2026] [UniProtKB: P06241]
ChEMBL	Dissociation constant for binding to SH2 domain of Fyn protein kinase	B	6.05	pKd	900	nM	Kd	J. Med. Chem. (1999) 42: 784-787 [PMID:10072676]
LCK proto-oncogene, Src family tyrosine kinase/Tyrosine-protein kinase LCK in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL258] [GtoPdb: 2053] [UniProtKB: P06239]
ChEMBL	Dissociation constant for binding to SH2 domain of p56 lck tyrosine kinase	B	5.89	pKd	1300	nM	Kd	J. Med. Chem. (1999) 42: 784-787 [PMID:10072676]
ChEMBL	Dissociation constant for binding to SH2 domain of p56 lck tyrosine kinase	B	6.19	pKd	640	nM	Kd	J. Med. Chem. (1999) 42: 784-787 [PMID:10072676]
FFA2 receptor in Human [GtoPdb: 226] [UniProtKB: O15552]
GtoPdb	-	-	4.6	pEC50	-	-	-	J Biol Chem (2003) 278: 11312-9 [PMID:12496283]; Biochem Biophys Res Commun (2003) 303: 1047-52 [PMID:12684041]; J Biol Chem (2003) 278: 25481-9 [PMID:12711604]; J Biol Chem (2011) 286: 10628-40 [PMID:21220428]

ChEMBL data shown on this page come from version 31:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]