compound 26 [PMID: 31710475] [Ligand Id: 10602] activity data from GtoPdb
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| mitogen-activated protein kinase kinase kinase 5 in Human [GtoPdb: 2080] [UniProtKB: Q99683] | ||||||||
| GtoPdb | Cellular assay; inhibition of ASK1-T838 autophosphorylation in HEK293T cells. | - | 6.83 | pIC50 | 148 | nM | IC50 | J Med Chem (2019) 62: 10740-10756 [PMID:31710475] |
| GtoPdb | Biochemical assay; inhibition of ASK1 autophosphorylation. | - | 8.22 | pIC50 | 6 | nM | IC50 | J Med Chem (2019) 62: 10740-10756 [PMID:31710475] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
