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ChEMBL ligand: CHEMBL1628548 (CGP-71872) |
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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GABAB2/GABAB1/GABA-B receptor in Human (target type: PROTEIN COMPLEX) [ChEMBL: CHEMBL2111463] [GtoPdb: 241, 240] [UniProtKB: O75899, Q9UBS5] | ||||||||
ChEMBL | Binding affinity to GABA-B receptor (unknown origin) | B | 9 | pKd | 1 | nM | Kd | J. Med. Chem. (2015) 58: 6336-6347 [PMID:25856547] |
GABAB2/GABAB1 in Rat [GtoPdb: 241, 240] [UniProtKB: O88871, Q9Z0U4] | ||||||||
GtoPdb | - | - | 9 | pKd | - | - | - | Nature (1997) 386: 239-46 [PMID:9069281] |
GABAB receptor in Rat [GtoPdb: 242] | ||||||||
GtoPdb | - | - | 9 | pKd | 1 | nM | Kd | Nature (1997) 386: 239-46 [PMID:9069281] |
ChEMBL data shown on this page come from version 31:
Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]