ChEMBL ligand: CHEMBL126 (Linezolid, Pnu-100766, U-100,766, U-100766, Zyvox)
DNA gyrase subunit A/DNA gyrase subunit B/DNA gyrase in Escherichia coli [ChEMBL: CHEMBL2094139] [GtoPdb: 3217, 3218] [UniProtKB: P0AES4, P0AES6] There should be some charts here, you may need to enable JavaScript!
Monoamine oxidase A in Human [ChEMBL: CHEMBL1951] [GtoPdb: 2489] [UniProtKB: P21397] There should be some charts here, you may need to enable JavaScript!
Monoamine oxidase B in Human [ChEMBL: CHEMBL2039] [GtoPdb: 2490] [UniProtKB: P27338] Monoamine oxidase B in Rat [ChEMBL: CHEMBL2993] [GtoPdb: 2490] [UniProtKB: P19643] There should be some charts here, you may need to enable JavaScript!
Succinate dehydrogenase [ubiquinone] flavoprotein subunit, mitochondrial in Human [ChEMBL: CHEMBL5758] [UniProtKB: P31040] There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
DNA gyrase subunit A/DNA gyrase subunit B/DNA gyrase in Escherichia coli (target type: PROTEIN COMPLEX) [ChEMBL: CHEMBL2094139] [GtoPdb: 3217, 3218] [UniProtKB: P0AES4, P0AES6]
ChEMBL	Inhibition of Escherichia coli DNA gyrase using fluorescence-tagged DNA by fluorescenct polarization assay	B	4.49	pIC50	>32000	nM	IC50	J Med Chem (2014) 57: 9078-9095 [PMID:25286019]
Monoamine oxidase A in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1951] [GtoPdb: 2489] [UniProtKB: P21397]
ChEMBL	Inhibition of monoamine oxidase A	B	4.26	pKi	55000	nM	Ki	J Med Chem (2008) 51: 1981-1990 [PMID:18338841]
ChEMBL	Inhibition of human recombinant MAOA	B	4.28	pKi	53000	nM	Ki	J Med Chem (2007) 50: 5886-5889 [PMID:17988109]
ChEMBL	Inhibition human liver MAOA activity	B	4.7	pKi	20000	nM	Ki	Bioorg Med Chem Lett (2007) 17: 337-340 [PMID:17095223]
ChEMBL	Inhibition of MAO-A (unknown origin) by luciferase reporter gene assay	B	5.1	pKi	7900	nM	Ki	Bioorg Med Chem (2013) 21: 577-591 [PMID:23273607]
ChEMBL	Reversible inhibition of human MAO-A	B	4.34	pIC50	46000	nM	IC50	Eur J Med Chem (2015) 106: 120-131 [PMID:26536532]
GtoPdb	-	-	4.34	pIC50	46000	nM	IC50	Eur J Med Chem (2015) 106: 120-31 [PMID:26536532]
Monoamine oxidase B in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2039] [GtoPdb: 2490] [UniProtKB: P27338]
ChEMBL	Inhibition of MAOB	B	4.77	pIC50	17000	nM	IC50	Eur J Med Chem (2009) 44: 3584-3590 [PMID:19321235]
ChEMBL	Reversible inhibition of human MAO-B	B	5.68	pIC50	2100	nM	IC50	Eur J Med Chem (2015) 106: 120-131 [PMID:26536532]
GtoPdb	-	-	5.68	pIC50	2100	nM	IC50	Eur J Med Chem (2015) 106: 120-31 [PMID:26536532]
GtoPdb	-	-	8.32	pIC50	4.77	nM	IC50	Eur J Med Chem (2009) 44: 3584-90 [PMID:19321235]
Monoamine oxidase B in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2993] [GtoPdb: 2490] [UniProtKB: P19643]
ChEMBL	Compound was evaluated for inhibition of Mono aminoxidase B in rat primary hepatocytes	B	4.77	pIC50	17000	nM	IC50	Bioorg Med Chem Lett (2002) 12: 2121-2123 [PMID:12127518]
Succinate dehydrogenase [ubiquinone] flavoprotein subunit, mitochondrial in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL5758] [UniProtKB: P31040]
ChEMBL	Inhibition of SDH-A (unknown origin) by ELISA	B	5.09	pIC50	8190	nM	IC50	Bioorg Med Chem Lett (2019) 29: 2686-2689 [PMID:31383589]

ChEMBL data shown on this page come from version 33:

Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]